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swapnil yerande
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Title
Cited by
Cited by
Year
2-Amino-5-thiazolyl motif: A novel scaffold for designing anti-inflammatory agents of diverse structures
PX Franklin, AD Pillai, PD Rathod, S Yerande, M Nivsarkar, H Padh, ...
European journal of medicinal chemistry 43 (1), 129-134, 2008
1242008
Syntheses of new tetrasubstituted thiophenes as novel anti-inflammatory agents
KI Molvi, KK Vasu, SG Yerande, V Sudarsanam, N Haque
European journal of medicinal chemistry 42 (8), 1049-1058, 2007
962007
Base-Mediated Hydroamination of Propargylamine: A Regioselective Intramolecular 5-exo-dig Cycloisomerization en Route to Imidazole-2-thione
A Ranjan, R Yerande, PB Wakchaure, SG Yerande, DH Dethe
Organic letters 16 (21), 5788-5791, 2014
752014
An asymmetric alkynylation/hydrothiolation cascade: an enantioselective synthesis of thiazolidine-2-imines from imines, acetylenes and isothiocyanates
A Ranjan, A Mandal, SG Yerande, DH Dethe
Chemical communications 51 (75), 14215-14218, 2015
462015
2-Amino-5-benzoyl-4-phenylthiazoles: Development of potent and selective adenosine A1 receptor antagonists
AB Scheiff, SG Yerande, A El-Tayeb, W Li, GS Inamdar, KK Vasu, ...
Bioorganic & Medicinal Chemistry 18 (6), 2195-2203, 2010
392010
Cyclization of active methylene isocyanides with α-oxodithioesters induced by base: An expedient synthesis of 4-methylthio/ethoxycarbonyl-5-acylthiazoles
KR Kiran, TR Swaroop, N Rajeev, SM Anil, KS Rangappa, MP Sadashiva
Synthesis 52 (09), 1444-1450, 2020
312020
Application of cyclic ketones in MCR: Ugi/amide coupling based synthesis of fused tetrazolo [1, 5-a][1, 4] benzodiazepines
SG Yerande, KM Newase, B Singh, A Boltjes, A Dömling
Tetrahedron letters 55 (21), 3263-3266, 2014
282014
Substituted 4-phenylthiazoles: Development of potent and selective A1, A3 and dual A1/A3 adenosine receptor antagonists
A Abdelrahman, SG Yerande, V Namasivayam, TA Klapschinski, ...
European Journal of Medicinal Chemistry 186, 111879, 2020
132020
Thiol–Yne Coupling of Propargylamine under Solvent‐Free Conditions by Bond Anion Relay Chemistry: An Efficient Synthesis of Thiazolidin‐2‐ylideneamine
A Ranjan, AS Deore, SG Yerande, DH Dethe
European Journal of Organic Chemistry 2017 (28), 4130-4139, 2017
122017
Efficient synthesis of indole derivatives containing the tetrazole moeity utilizing an Ugi-Azide post-transformation strategy
A Nikbakht, S Balalaie, F Baghestani, F Rominger
Synlett 29 (14), 1892-1896, 2018
102018
Activation of Primary Amines by Copper (I)-Based Lewis Acid Promoters in the Solventless Synthesis of Secondary Propargylamines
C Cimarelli, F Navazio, FV Rossi, F Del Bello, E Marcantoni
Synthesis 51 (11), 2387-2396, 2019
62019
Thiazole and thiophene analogues, and their use in treating autoimmune diseases and cancers
A Giordano, KK Vasu, HM Thakar, RS Giri, SG Yerande, GS Inamdar, ...
US Patent 8,217,037, 2012
62012
Fries rearrangement: scalable synthesis of key fluoro building blocks 3-fluoro-4-methoxybenzoyl chloride and 1, 2-diethoxy-3-fluorobenzene
SG Yerande, DM Shendage, PB Wakchaure, GR Phadtare, MY Bhoite, ...
Tetrahedron letters 55 (15), 2426-2429, 2014
52014
Synthesis, antiinflammatory and HIV-1 integrase inhibitory activities of 1, 2-bis [5-thiazolyl] ethane-1, 2-dione derivatives
PX Franklin, S Yerande, HM Thakar, GS Inamdar, RS Giri, H Padh, ...
Indian journal of pharmaceutical sciences 71 (3), 259, 2009
52009
WO 2006148113, 2007
V Sudarsanam, A Giordano, KK Vasu, HM Thakar, RS Giri, S Yerande, ...
Chem. Abstr 147, 469324, 2007
52007
Mercury (II) Chloride‐Mediated Desulphurization of Amidinothioureas: Synthesis and Antimicrobial Activity of 3‐Amino‐1, 2, 4‐triazole Derivatives
SG Yerande, CD Baviskar, KM Newase, W Wang, K Wang, A Dömling
Journal of Heterocyclic Chemistry 51 (6), 1883-1887, 2014
42014
(3+ 2) Annulation of Amidinothioureas with Binucleophile: Synthesis and Antimicrobial Activity of 3‐Phenylamino‐5‐aryl/alkyl‐1, 2, 4‐oxadiazole Derivatives
SG Yerande, AB Ghaisas, KM Newase, W Wang, K Wang, A Doemling
Journal of Heterocyclic Chemistry 51 (6), 1752-1756, 2014
42014
A Facile Diversity‐Oriented Multicomponent One‐Pot Synthesis of 3‐Amino‐6,7‐dihydrobenzo[c]thiophen‐4(5H)‐one Derivatives from α‐Oxo‐N,S‐ketene Acetal
SG Yerande, SD More, M Bhandari, KM Newase, K Khoury, K Wang, ...
Journal of Heterocyclic Chemistry 51 (S1), E358-E363, 2014
42014
A Method for the Racemization of 2-Methylpyrrolidine: A Histamine H3 Receptor Pharmacophore
SG Yerande, RS Yerande, PP Thakare, DM Shendage, S Galave, ...
Organic Process Research & Development 18 (5), 652-655, 2014
42014
One‐Pot Synthesis of 2‐Amino‐1, 3‐selenazole via an Intermediary Amidinoselenourea
A Ranjan, R Yerande, M Jadhav, SG Yerande, DH Dethe
European Journal of Organic Chemistry 2015 (15), 3230-3234, 2015
22015
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