| Novel N-indolylmethyl substituted olanzapine derivatives: their design, synthesis and evaluation as PDE4B inhibitors DR Gorja, S Mukherjee, CLT Meda, GS Deora, KL Kumar, A Jain, ... Organic & Biomolecular Chemistry 11 (13), 2075-2079, 2013 | 71 | 2013 |
| Oral dosing in adult zebrafish: proof-of-concept using pharmacokinetics and pharmacological evaluation of carbamazepine P Kulkarni, GH Chaudhari, V Sripuram, RK Banote, KT Kirla, R Sultana, ... Pharmacological Reports 66, 179-183, 2014 | 63 | 2014 |
| Design and synthesis of novel quinoline–aminopiperidine hybrid analogues as Mycobacterium tuberculosis DNA gyraseB inhibitors B Medapi, J Renuka, S Saxena, JP Sridevi, R Medishetti, P Kulkarni, ... Bioorganic & medicinal chemistry 23 (9), 2062-2078, 2015 | 58 | 2015 |
| Larval zebrafish model for studying the effects of valproic acid on neurodevelopment: An approach towards modeling autism S Dwivedi, R Medishetti, R Rani, A Sevilimedu, P Kulkarni, P Yogeeswari Journal of pharmacological and toxicological methods 95, 56-65, 2019 | 56 | 2019 |
| 5-Benzylidene-2, 4-thiazolidenedione derivatives: Design, synthesis and evaluation as inhibitors of angiogenesis targeting VEGR-2 U Bhanushali, S Rajendran, K Sarma, P Kulkarni, K Chatti, S Chatterjee, ... Bioorganic chemistry 67, 139-147, 2016 | 56 | 2016 |
| Optimization of the adult zebrafish ECG method for assessment of drug-induced QTc prolongation GH Chaudhari, KS Chennubhotla, K Chatti, P Kulkarni Journal of pharmacological and toxicological methods 67 (2), 115-120, 2013 | 55 | 2013 |
| Distribution of BDE-99 and effects on metamorphosis of BDE-99 and-47 after oral exposure in Xenopus tropicalis G Carlsson, P Kulkarni, P Larsson, L Norrgren Aquatic toxicology 84 (1), 71-79, 2007 | 51 | 2007 |
| AlCl 3-mediated hydroarylation–heteroarylation in a single pot: a direct access to densely functionalized olefins of pharmacological interest A Nakhi, S Archana, GPK Seerapu, KS Chennubhotla, KL Kumar, ... Chemical communications 49 (56), 6268-6270, 2013 | 44 | 2013 |
| Oral gabapentin suppresses pentylenetetrazole-induced seizure-like behavior and cephalic field potential in adult zebrafish RK Banote, S Koutarapu, KS Chennubhotla, K Chatti, P Kulkarni Epilepsy & Behavior 27 (1), 212-219, 2013 | 41 | 2013 |
| Novel zebrafish EAE model: A quick in vivo screen for multiple sclerosis P Kulkarni, S Yellanki, R Medishetti, D Sriram, U Saxena, P Yogeeswari Multiple sclerosis and related disorders 11, 32-39, 2017 | 31 | 2017 |
| Development of novel N-linked aminopiperidine-based mycobacterial DNA gyrase B inhibitors: scaffold hopping from known antibacterial leads VU Jeankumar, J Renuka, VK Pulla, V Soni, JP Sridevi, P Suryadevara, ... International journal of antimicrobial agents 43 (3), 269-278, 2014 | 31 | 2014 |
| Development of acridine derivatives as selective Mycobacterium tuberculosis DNA gyrase inhibitors B Medapi, N Meda, P Kulkarni, P Yogeeswari, D Sriram Bioorganic & medicinal chemistry 24 (4), 877-885, 2016 | 30 | 2016 |
| Transition metal free hydrolysis/cyclization strategy in a single pot: synthesis of fused furo N-heterocycles of pharmacological interest A Nakhi, MS Rahman, GPK Seerapu, RK Banote, KL Kumar, P Kulkarni, ... Organic & Biomolecular Chemistry 11 (30), 4930-4934, 2013 | 29 | 2013 |
| Structure-guided design and development of novel benzimidazole class of compounds targeting DNA gyraseB enzyme of Staphylococcus aureus R Janupally, VU Jeankumar, KA Bobesh, V Soni, PB Devi, VK Pulla, ... Bioorganic & Medicinal Chemistry 22 (21), 5970-5987, 2014 | 28 | 2014 |
| Ligand/PTC-free intramolecular Heck reaction: synthesis of pyrroloquinoxalines and their evaluation against PDE4/luciferase/oral cancer cell growth in vitro and zebrafish in vivo PV Babu, S Mukherjee, GS Deora, KS Chennubhotla, R Medisetti, ... Organic & Biomolecular Chemistry 11 (39), 6680-6685, 2013 | 28 | 2013 |
| InCl3 mediated heteroarylation of indoles and their derivatization via CH activation strategy: Discovery of 2-(1H-indol-3-yl)-quinoxaline derivatives as a new class of PDE4B … R Sunke, R Bankala, B Thirupataiah, EVVS Ramarao, JS Kumar, ... European Journal of Medicinal Chemistry 174, 198-215, 2019 | 27 | 2019 |
| Exploring the gyrase ATPase domain for tailoring newer anti-tubercular drugs: hit to lead optimization of a novel class of thiazole inhibitors VU Jeankumar, S Kotagiri, R Janupally, P Suryadevara, JP Sridevi, ... Bioorganic & Medicinal Chemistry 23 (3), 588-601, 2015 | 26 | 2015 |
| Optimization and validation of Mycobacterium marinum-induced adult zebrafish model for evaluation of oral anti-tuberculosis drugs JP Sridevi, HS Anantaraju, P Kulkarni, P Yogeeswari, D Sriram The International Journal of Mycobacteriology 3 (4), 259-267, 2014 | 26 | 2014 |
| Enabling the (3+ 2) cycloaddition reaction in assembling newer anti-tubercular lead acting through the inhibition of the gyrase ATPase domain: lead optimization and structure … VU Jeankumar, RS Reshma, R Janupally, S Saxena, JP Sridevi, ... Organic & Biomolecular Chemistry 13 (8), 2423-2431, 2015 | 25 | 2015 |
| NaSH in the construction of thiophene ring fused with N-heterocycles: A rapid and inexpensive synthesis of novel small molecules as potential inducers of apoptosis SK Kolli, A Nakhi, R Medishetti, S Yellanki, P Kulkarni, RR Raju, M Pal Bioorganic & Medicinal Chemistry Letters 24 (18), 4460-4465, 2014 | 21 | 2014 |
Raghavender MedishettyDr.Reddys institiute of life sciencesVerified email at drils.org
