Discovery of certain benzyl/phenethyl thiazolidinone-indole hybrids as potential anti-proliferative agents: Synthesis, molecular modeling and tubulin polymerization inhibition … DK Sigalapalli, V Pooladanda, P Singh, M Kadagathur, SD Guggilapu, ... Bioorganic chemistry 92, 103188, 2019 | 35 | 2019 |
Novel diindoloazepinone derivatives as DNA minor groove binding agents with selective topoisomerase I inhibition: Design, synthesis, biological evaluation and docking studies M Kadagathur, GP Devi, P Grewal, DK Sigalapalli, PN Makhal, ... Bioorganic Chemistry 99, 103629, 2020 | 29 | 2020 |
Facile synthesis of 2-aryl 5-hydroxy benzo [d] oxazoles and their in vitro anti-proliferative effects on various cancer cell lines ND Tangellamudi, SB Shinde, V Pooladanda, C Godugu, ... Bioorganic & Medicinal Chemistry Letters 28 (23-24), 3639-3647, 2018 | 19 | 2018 |
Synthesis and biological evaluation of novel imidazo [1, 2-a] pyridine-oxadiazole hybrids as anti-proliferative agents: Study of microtubule polymerization inhibition and DNA … DK Sigalapalli, G Kiranmai, GP Devi, R Tokala, S Sana, C Tripura, ... Bioorganic & Medicinal Chemistry 43, 116277, 2021 | 16 | 2021 |
Novel chromenyl-based 2-iminothiazolidin-4-one derivatives as tubulin polymerization inhibitors: Design, synthesis, biological evaluation and molecular modelling studies DK Sigalapalli, V Pooladanda, M Kadagathur, SD Guggilapu, JL Uppu, ... Journal of Molecular Structure 1225, 128847, 2021 | 16 | 2021 |
Sequential C–N and C–O Bond Formation in a Single Pot: Synthesis of 2H-Benzo[b][1,4]oxazines from 2,5-Dihydroxybenzaldehyde and Amino acid Precursors J Iqbal, ND Tangellamudi, B Dulla, S Balasubramanian Organic letters 14 (2), 552-555, 2012 | 16 | 2012 |
Synthesis of indolo/pyrroloazepinone-oxindoles as potential cytotoxic, DNA-intercalating and Topo I inhibitors M Kadagathur, AS Shaikh, B Panda, J George, R Phanindranath, ... Bioorganic Chemistry 122, 105706, 2022 | 15 | 2022 |
Isovanillin derived N-(un) substituted hydroxylamines possessing an ortho-allylic group: valuable precursors to bioactive N-heterocycles B Dulla, ND Tangellamudi, S Balasubramanian, S Yellanki, R Medishetti, ... Organic & Biomolecular Chemistry 12 (16), 2552-2558, 2014 | 15 | 2014 |
Targeting tubulin polymerization and DNA binding of 4-thiazolidinone–umbelliferone hybrids: synthesis and cytotoxicity evaluation DK Sigalapalli, G Kiranmai, R Tokala, C Tripura, R Ambatwar, ... New Journal of Chemistry 45 (40), 18908-18923, 2021 | 12 | 2021 |
Exploration of mercaptoacetamide-linked pyrimidine-1, 3, 4-oxadiazole derivatives as DNA intercalative topo II inhibitors: Cytotoxicity and apoptosis induction AS Shaikh, G Kiranmai, GP Devi, PN Makhal, DK Sigalapalli, R Tokala, ... Bioorganic & Medicinal Chemistry Letters 65, 128697, 2022 | 11 | 2022 |
Design, synthesis of DNA-interactive 4-thiazolidinone-based indolo-/pyrroloazepinone conjugates as potential cytotoxic and topoisomerase I inhibitors M Kadagathur, S Patra, G Devabattula, J George, R Phanindranath, ... European Journal of Medicinal Chemistry 238, 114465, 2022 | 10 | 2022 |
Cyclodesulfurization: an enabling protocol for synthesis of various heterocycles M Kadagathur, AS Shaikh, GS Jadhav, DK Sigalapalli, N Shankaraiah, ... ChemistrySelect 6 (10), 2621-2640, 2021 | 10 | 2021 |
Syntheses and medicinal chemistry of azepinoindolones: a look back to leap forward M Kadagathur, S Patra, DK Sigalapalli, N Shankaraiah, ND Tangellamudi Organic & Biomolecular Chemistry 19 (4), 738-764, 2021 | 10 | 2021 |
Microwave-assisted hydrogen peroxide-mediated synthesis of benzoxazoles and related heterocycles via cyclodesulfurization M Kadagathur, DK Sigalapalli, S Patra, ND Tangellamudi Synthetic Communications 51 (14), 2213-2224, 2021 | 8 | 2021 |
Novel Huperzine A based NMDA antagonists: Insights from Molecular Docking, ADME/T and Molecular Dynamics Simulation Studies RR DILEP SIGALAPALLI, NEELIMA D. TANGELLAMUDI RSC ADVANCES 10, 25446-25455, 2020 | 7 | 2020 |
Quinacetophenone: A Simple Precursor for Synthesis of Phenoxazines NDT Saiprasad N. Nunewar,Bhavana B. Muthyala, Sowmya Dastari New Journal of Chemistry, 2019 | 6 | 2019 |
Insights into the pharmacophore-based 3D-QSAR modeling, molecular dynamics simulation studies of certain dihydroxy pyrrolidine/piperidine and aza-flavanone derivatives as α … DK Sigalapalli, V Yele, S Jupudi, AS Shaikh, M Kadagathur, ... Journal of Molecular Structure 1223, 129243, 2021 | 5 | 2021 |
Synthesis of 1-(Indol-2-yl)-phenoxazine hybrids from quinacetophenone precursors and their biological evaluation as DNA intercalating agents SN Nunewar, N Kotla, JL Uppu, A Dixit, V Pooladanda, C Godugu, ... Journal of Molecular Structure 1217, 128311, 2020 | 5 | 2020 |
Unexpected chemoselectivity of cyclic enones on introducing additional chirality in diethanolamine ligand in catalytic asymmetric Michael addition reactions using heterobimetallics ND Tangellamudi, S Govindarajan Journal of Molecular Catalysis A: Chemical 314 (1-2), 71-80, 2009 | 4 | 2009 |
Microwave‐Assisted TBHP‐Mediated Synthesis of 2‐Amino‐1, 3, 4‐oxadiazoles in Water D Kumar Sigalapalli, M Kadagathur, A Sujat Shaikh, GS Jadhav, B Bakchi, ... ChemistrySelect 5 (42), 13248-13258, 2020 | 3 | 2020 |