Practical Alkoxythiocarbonyl Auxiliaries for Ir(I)-Catalyzed C-H Alkylation of Azacycles AT Tran, JQ Yu Angew. Chem. int. Ed. 56 (35), 10530-10534, 2017 | 97* | 2017 |
Identification of selective inhibitors of indoleamine 2, 3-dioxygenase 2 SM Bakmiwewa, AA Fatokun, A Tran, RJ Payne, NH Hunt, HJ Ball Bioorganic & medicinal chemistry letters 22 (24), 7641-7646, 2012 | 61 | 2012 |
Sansanmycin natural product analogues as potent and selective anti-mycobacterials that inhibit lipid I biosynthesis AT Tran, EE Watson, V Pujari, T Conroy, LJ Dowman, AM Giltrap, A Pang, ... Nature communications 8 (1), 14414, 2017 | 54 | 2017 |
Discovery of potent and selective non-nucleotide small molecule inhibitors of CD73 JW Beatty, EA Lindsey, R Thomas-Tran, L Debien, D Mandal, JL Jeffrey, ... Journal of medicinal chemistry 63 (8), 3935-3955, 2020 | 40 | 2020 |
Inhibition studies on Mycobacterium tuberculosis N-acetylglucosamine-1-phosphate uridyltransferase (GlmU) AT Tran, D Wen, NP West, EN Baker, WJ Britton, RJ Payne Organic & biomolecular chemistry 11 (46), 8113-8126, 2013 | 34 | 2013 |
β-C(sp3)–H Arylation of α-Hydroxy Acid Derivatives Utilizing Amino Acid as a Directing Group T Tetsuya, Y Hu, AT Tran, JQ Yu Org. Lett. 17 (24), 5966-5969, 2015 | 33 | 2015 |
Elucidation of Mycobacterium tuberculosis Type II Dehydroquinase Inhibitors using a Fragment Elaboration Strategy AT Tran, NP West, WJ Britton, RJ Payne ChemMedChem 7 (6), 1031-1043, 2012 | 26 | 2012 |
Rapid assembly of potent type II dehydroquinase inhibitors via “Click” chemistry AT Tran, KM Cergol, WJ Britton, SAI Bokhari, M Ibrahim, AJ Lapthorn, ... MedChemComm 1 (4), 271-275, 2010 | 23 | 2010 |
Synthesis and evaluation of potent ene-yne inhibitors of type II dehydroquinases as tuberculosis drug leads AT Tran, KM Cergol, NP West, EJ Randall, WJ Britton, SAI Bokhari, ... ChemMedChem 6 (2), 262-265, 2011 | 16 | 2011 |
Development of a Scalable Method for Manufacturing the Central Core of CD73 Inhibitor AB680 J Fournier, X Yan, AT Tran, RL Grange, SD Jacob, J Kalisiak, KV Lawson, ... Organic Process Research & Development 25 (1), 157-162, 2020 | 5 | 2020 |
Practical alkoxythiocarbonyl auxiliaries for Ir (I)-catalyzed Cu2013H hydroalkylation of azacycles J Yu, AT Tran American Chemical Society SciMeetings 1 (2), 2020 | | 2020 |
Preparation of substituted 1-amino-2-[3-(dihydroxyboranyl)propyl]-2,3- dihydro-1H-indene-1-carboxylic acids as inhibitors of ARG1 and/or ARG2 J Beatty, CN Foley, RL Grange, T Guney, SD Jacob, J Kalisiak, MR Leleti, ... US Patent WO2,020,102,646, 2020 | | 2020 |
Heterobicyclic compounds as CD73 inhibitors and their preparation J Beatty, LPP Debien, SL Drew, J Fournier, RL Grange, SD Jacob, ... US Patent WO2,020,046,813, 2020 | | 2020 |
Arginase inhibitors CN Foley, RL Grange, T Guney, J Kalisiak, ET Newcomb, AT Tran US Patent WO2,019,173,188, 2019 | | 2019 |
Preparation of nucleosidyl peptides, including sansanmycin analogs, as anti-mycobacterials RJ Payne, WJ Britton, A Tran, W Tran AU Patent WO2,018,107,236, 2018 | | 2018 |
β-C (sp3) â H Arylation of α-Hydroxy Acid Derivatives Utilizing Amino Acid as a Directing Group T Toba, Y Hu, AT Tran, JQ Yu Organic letters 17 (24), 2015 | | 2015 |