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Dr. Suyog M. Amrutkar
Dr. Suyog M. Amrutkar
Verified email at niper.ac.in
Title
Cited by
Cited by
Year
Switch in site of inhibition: a strategy for structure-based discovery of human topoisomerase IIα catalytic inhibitors
AT Baviskar, SM Amrutkar, N Trivedi, V Chaudhary, A Nayak, SK Guchhait, ...
ACS medicinal chemistry letters 6 (4), 481-485, 2015
992015
Imine/amide–imidazole conjugates derived from 5-amino-4-cyano-N1-substituted benzyl imidazole: Microwave-assisted synthesis and anticancer activity via …
A Negi, JM Alex, SM Amrutkar, AT Baviskar, G Joshi, S Singh, ...
Bioorganic & medicinal chemistry 23 (17), 5654-5661, 2015
532015
Scaffold-hopping of bioactive flavonoids: Discovery of aryl-pyridopyrimidinones as potent anticancer agents that inhibit catalytic role of topoisomerase IIα
G Priyadarshani, S Amrutkar, A Nayak, UC Banerjee, CN Kundu, ...
European Journal of Medicinal Chemistry 122, 43-54, 2016
392016
Scaffold-Hopping of Aurones: 2-Arylideneimidazo[1,2-a]pyridinones as Topoisomerase IIα-Inhibiting Anticancer Agents
G Priyadarshani, A Nayak, SM Amrutkar, S Das, SK Guchhait, CN Kundu, ...
ACS Medicinal Chemistry Letters 7 (12), 1056-1061, 2016
362016
Dual inhibitors of epidermal growth factor receptor and topoisomerase IIα derived from a quinoline scaffold
M Chauhan, G Joshi, H Kler, A Kashyap, SM Amrutkar, P Sharma, ...
RSC advances 6 (81), 77717-77734, 2016
322016
Synthesis and biological evaluation of new 2, 5-dimethylthiophene/furan based N-acetyl pyrazolines as selective topoisomerase II inhibitors
G Joshi, SM Amrutkar, AT Baviskar, H Kler, S Singh, UC Banerjee, ...
RSC advances 6 (18), 14880-14892, 2016
262016
E-pharmacophore guided discovery of pyrazolo [1, 5-c] quinazolines as dual inhibitors of topoisomerase-I and histone deacetylase
G Joshi, S Kalra, UP Yadav, P Sharma, PK Singh, S Amrutkar, AJ Ansari, ...
Bioorganic Chemistry 94, 103409, 2020
252020
One-pot synthesis of (R)-1-(1-naphthyl) ethanol by stereoinversion using Candida parapsilosis
SM Amrutkar, L Banoth, UC Banerjee
Tetrahedron Letters 54 (25), 3274-3277, 2013
212013
Anticancer activity of dihydropyrazolo[1,5‐c]quinazolines against rat C6 glioma cells via inhibition of topoisomerase II
G Kaur, RP Cholia, G Joshi, SM Amrutkar, S Kalra, AK Mantha, ...
Archiv der Pharmazie 351 (6), 1800023, 2018
122018
Sulfinate based selective labelling of 5-hydroxy methylcytosine: Application to biotin pull down assay
W Qiong, SM Amrutkar, F Shao
Bioconjugate chemistry 29 (2), 245-249, 2018
112018
Chapter 3.TARGETING HUMAN TOPOISOMERASE-II: OPPORTUNITIES IN CANCER CHEMOTHERAPY
SM Amrutkar, KD Bhilare
Topoisomerase Inhibitors: Classification, Mechanisms of Action and Adverse …, 2017
2017
Structure based design with modulation of known ligands leading to switch in mode of inhibition of human topoisomerase II alpha
S Amrutkar, S Guchhait, U Banerjee
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 251, 2016
2016
Dual inhibitors of epidermal growth factor receptor and topoisomerase IIa derived from a quinoline scaffold
M Chauhan, G Joshi, H Kler, A Kashyap, SM Amrutkar, P Sharma, ...
Royal Society of Chemistry, 2016
2016
Establishment of a strategy," choice based change", in mode of inhibition: Development of imidazo [1, 2-a] pyridines/pyrazines as novel topoisomerase II alpha catalytic inhibitors
S Amrutkar, S Guchhait, U Banerjee
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 250, 2015
2015
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