| Discovery of new quinolines as potent colchicine binding site inhibitors: Design, synthesis, docking studies, and anti-proliferative evaluation M Hagras, MA El Deeb, HSA Elzahabi, EB Elkaeed, ABM Mehany, ... Journal of enzyme inhibition and medicinal chemistry 36 (1), 640-658, 2021 | 58 | 2021 |
| Arylthiazole antibiotics targeting intracellular methicillin-resistant Staphylococcus aureus (MRSA) that interfere with bacterial cell wall synthesis I Eid, MM Elsebaei, H Mohammad, M Hagras, CE Peters, YA Hegazy, ... European journal of medicinal chemistry 139, 665-673, 2017 | 49 | 2017 |
| Medicinal attributes of pyridine scaffold as anticancer targeting agents EA Mohamed, NSM Ismail, M Hagras, H Refaat Future Journal of Pharmaceutical Sciences 7, 1-17, 2021 | 46 | 2021 |
| Investigating the Antibacterial Activity of Biphenylthiazoles against Methicillin- and Vancomycin-Resistant Staphylococcus aureus (MRSA and VRSA) M Hagras, H Mohammad, MS Mandour, YA Hegazy, A Ghiaty, ... Journal of Medicinal Chemistry 60 (9), 4074-4085, 2017 | 45 | 2017 |
| Phenylthiazoles with tert-Butyl side chain: Metabolically stable with anti-biofilm activity A Kotb, NS Abutaleb, MA Seleem, M Hagras, H Mohammad, A Bayoumi, ... European journal of medicinal chemistry 151, 110-120, 2018 | 43 | 2018 |
| Synthesis and antibacterial evaluation of a novel library of 2-(thiazol-5-yl)-1, 3, 4-oxadiazole derivatives against methicillin-resistant Staphylococcus aureus (MRSA) MH Hannoun, M Hagras, A Kotb, AAMM El-Attar, HS Abulkhair Bioorganic chemistry 94, 103364, 2020 | 42 | 2020 |
| Discovery of pyrazolo [3, 4-d] pyrimidine and pyrazolo [4, 3-e][1, 2, 4] triazolo [1, 5-c] pyrimidine derivatives as novel CDK2 inhibitors: synthesis, biological and molecular … IF Nassar, MTA Aal, WA El-Sayed, MAE Shahin, EGE Elsakka, ... RSC advances 12 (23), 14865-14882, 2022 | 34 | 2022 |
| 1,3,4-Oxadiazole-naphthalene hybrids as potential VEGFR-2 inhibitors: design, synthesis, antiproliferative activity, apoptotic effect, and in silico studies M Hagras, MA Saleh, RR Ezz Eldin, AA Abuelkhir, EG Khidr, ... Journal of enzyme inhibition and medicinal chemistry 37 (1), 386-402, 2022 | 33 | 2022 |
| Naphthylthiazoles: Targeting Multidrug-Resistant and Intracellular Staphylococcus aureus with Biofilm Disruption Activity M Hagras, NS Abutaleb, AO Ali, JA Abdel-Aleem, MM Elsebaei, ... ACS infectious diseases 4 (12), 1679-1691, 2018 | 30 | 2018 |
| Biphenylthiazole antibiotics with an oxadiazole linker: An approach to improve physicochemical properties and oral bioavailability M Hagras, YA Hegazy, AH Elkabbany, H Mohammad, A Ghiaty, ... European journal of medicinal chemistry 143, 1448-1456, 2018 | 28 | 2018 |
| Alkoxyphenylthiazoles with broad-spectrum activity against multidrug-resistant gram-positive bacterial pathogens M ElAwamy, H Mohammad, A Hussien, NS Abutaleb, M Hagras, ... European Journal of Medicinal Chemistry 152, 318-328, 2018 | 27 | 2018 |
| Development of pyrolo [2, 3-c] pyrazole, pyrolo [2, 3-d] pyrimidine and their bioisosteres as novel CDK2 inhibitors with potent in vitro apoptotic anti-proliferative activity … EM Azmy, M Hagras, MA Ewida, AS Doghish, EG Khidr, AA El-Husseiny, ... Bioorganic Chemistry 139, 106729, 2023 | 24 | 2023 |
| Oxadiazolylthiazoles as novel and selective antifungal agents M Hagras, EA Salama, AM Sayed, NS Abutaleb, A Kotb, MN Seleem, ... European journal of medicinal chemistry 189, 112046, 2020 | 24 | 2020 |
| Synthesis, biological evaluation, and in silico studies of new CDK2 inhibitors based on pyrazolo [3, 4-d] pyrimidine and pyrazolo [4, 3-e][1, 2, 4] triazolo [1, 5-c] pyrimidine … AA Mandour, IF Nassar, MT Abdel Aal, MAE Shahin, WA El-Sayed, ... Journal of enzyme inhibition and medicinal chemistry 37 (1), 1957-1973, 2022 | 21 | 2022 |
| Synthesis, characterization and antimicrobial evaluation of some novel quinoline derivatives bearing different heterocyclic moieties KM El-Gamal, MS Hagrs, HS Abulkhair Bulletin of Faculty of Pharmacy, Cairo University 54 (2), 263-273, 2016 | 21 | 2016 |
| Design, synthesis, and anti-cancer evaluation of new pyrido [2, 3-d] pyrimidin-4 (3H)-one derivatives as potential EGFRWT and EGFRT790M inhibitors and apoptosis inducers HSA Elzahabi, ES Nossier, RA Alasfoury, M El-Manawaty, SM Sayed, ... Journal of Enzyme Inhibition and Medicinal Chemistry 37 (1), 1053-1076, 2022 | 18 | 2022 |
| Phenylthiazoles with nitrogenous side chain: An approach to overcome molecular obesity MM Elsebaei, NS Abutaleb, AA Mahgoub, D Li, M Hagras, H Mohammad, ... European Journal of Medicinal Chemistry 182, 111593, 2019 | 18 | 2019 |
| tert-Butylphenylthiazoles with an oxadiazole linker: a novel orally bioavailable class of antibiotics exhibiting antibiofilm activity A Kotb, NS Abutaleb, M Hagras, A Bayoumi, MM Moustafa, A Ghiaty, ... RSC advances 9 (12), 6770-6778, 2019 | 18 | 2019 |
| Development of Biphenylthiazoles Exhibiting Improved Pharmacokinetics and Potent Activity Against Intracellular Staphylococcus aureus M Hagras, NS Abutaleb, NM Elhosseiny, TM Abdelghany, M Omara, ... ACS Infectious Diseases 6 (11), 2887-2900, 2020 | 13 | 2020 |
| Design, Synthesis, biological Evaluation, and molecular docking studies of novel Pyrazolo [3, 4-d] Pyrimidine derivative scaffolds as potent EGFR inhibitors and cell apoptosis … FF Sherbiny, AH Bayoumi, AM El-Morsy, M Sobhy, M Hagras Bioorganic Chemistry 116, 105325, 2021 | 12 | 2021 |
Abdelrahman S. MayhoubProfessor, Zewail City for Science and TechnologyVerified email at zewailcity.edu.eg
