| Gamma‐glutamyl transpeptidase substrate specificity and catalytic mechanism JW Keillor, R Castonguay, C Lherbet Methods in enzymology 401, 449-467, 2005 | 126 | 2005 |
| Synthesis and biological activities of triazole derivatives as inhibitors of InhA and antituberculosis agents C Menendez, S Gau, C Lherbet, F Rodriguez, C Inard, MR Pasca, ... European journal of medicinal chemistry 46 (11), 5524-5531, 2011 | 118 | 2011 |
| Chemical synthesis and biological evaluation of triazole derivatives as inhibitors of InhA and antituberculosis agents C Menendez, A Chollet, F Rodriguez, C Inard, MR Pasca, C Lherbet, ... European journal of medicinal chemistry 52, 275-283, 2012 | 106 | 2012 |
| Synthesis, antimycobacterial screening and ligand-based molecular docking studies on novel pyrrole derivatives bearing pyrazoline, isoxazole and phenyl thiourea moieties SD Joshi, SR Dixit, MN Kirankumar, TM Aminabhavi, K Raju, R Narayan, ... European journal of medicinal chemistry 107, 133-152, 2016 | 96 | 2016 |
| Mechanochemical synthesis and biological evaluation of novel isoniazid derivatives with potent antitubercular activity PFM Oliveira, B Guidetti, A Chamayou, C André-Barrès, J Madacki, ... Molecules 22 (9), 1457, 2017 | 82 | 2017 |
| Design, chemical synthesis of 3-(9H-fluoren-9-yl) pyrrolidine-2, 5-dione derivatives and biological activity against enoyl-ACP reductase (InhA) and Mycobacterium tuberculosis T Matviiuk, F Rodriguez, N Saffon, S Mallet-Ladeira, M Gorichko, ... European Journal of Medicinal Chemistry 70, 37-48, 2013 | 55 | 2013 |
| Synthesis, characterization and antitubercular activities of novel pyrrolyl hydrazones and their Cu-complexes SD Joshi, D Kumar, SR Dixit, N Tigadi, UA More, C Lherbet, ... European journal of medicinal chemistry 121, 21-39, 2016 | 53 | 2016 |
| Design, synthesis and evaluation of new GEQ derivatives as inhibitors of InhA enzyme and Mycobacterium tuberculosis growth A Chollet, G Mori, C Menendez, F Rodriguez, I Fabing, MR Pasca, ... European Journal of Medicinal Chemistry 101, 218-235, 2015 | 50 | 2015 |
| Synthesis of 3-heteryl substituted pyrrolidine-2, 5-diones via catalytic Michael reaction and evaluation of their inhibitory activity against InhA and Mycobacterium tuberculosis T Matviiuk, G Mori, C Lherbet, F Rodriguez, MR Pasca, M Gorichko, ... European Journal of Medicinal Chemistry 71, 46-52, 2014 | 50 | 2014 |
| An overview on crystal structures of InhA protein: Apo-form, in complex with its natural ligands and inhibitors A Chollet, L Maveyraud, C Lherbet, V Bernardes-Génisson European journal of medicinal chemistry 146, 318-343, 2018 | 49 | 2018 |
| Crystal structure of the enoyl-ACP reductase of Mycobacterium tuberculosis (InhA) in the apo-form and in complex with the active metabolite of isoniazid pre-formed by a … A Chollet, L Mourey, C Lherbet, A Delbot, S Julien, M Baltas, J Bernadou, ... Journal of structural biology 190 (3), 328-337, 2015 | 49 | 2015 |
| Kinetic characterization and identification of the acylation and glycosylation sites of recombinant human γ-glutamyltranspeptidase R Castonguay, D Halim, M Morin, A Furtos, C Lherbet, E Bonneil, ... Biochemistry 46 (43), 12253-12262, 2007 | 43 | 2007 |
| Pyrrolidinone and pyrrolidine derivatives: Evaluation as inhibitors of InhA and Mycobacterium tuberculosis T Matviiuk, J Madacki, G Mori, BS Orena, C Menendez, A Kysil, ... European Journal of Medicinal Chemistry 123, 462-475, 2016 | 39 | 2016 |
| Cell permeation of a Trypanosoma brucei aldolase inhibitor: evaluation of different enzyme-labile phosphate protecting groups L Azéma, C Lherbet, C Baudoin, C Blonski Bioorganic & medicinal chemistry letters 16 (13), 3440-3443, 2006 | 36 | 2006 |
| Probing the stereochemistry of the active site of gamma-glutamyl transpeptidase using sulfur derivatives of l-glutamic acid C Lherbet, JW Keillor Organic & Biomolecular Chemistry 2 (2), 238-245, 2004 | 36 | 2004 |
| Synthesis and evaluation of α-ketotriazoles and α, β-diketotriazoles as inhibitors of Mycobacterium tuberculosis C Menendez, F Rodriguez, ALJL Ribeiro, F Zara, C Frongia, V Lobjois, ... European Journal of Medicinal Chemistry 69, 167-173, 2013 | 33 | 2013 |
| Cloning and expression of IspDF from Mesorhizobium loti. Characterization of a bifunctional protein that catalyzes non-consecutive steps in the methylerythritol phosphate pathway CA Testa, C Lherbet, F Pojer, JP Noel, CD Poulter Biochimica et Biophysica Acta (BBA)-Proteins and Proteomics 1764 (1), 85-96, 2006 | 33 | 2006 |
| Kinetic studies of rat kidney γ-glutamyltranspeptidase deacylation reveal a general base-catalyzed mechanism R Castonguay, C Lherbet, JW Keillor Biochemistry 42 (39), 11504-11513, 2003 | 33 | 2003 |
| Design and synthesis of thiourea-based derivatives as Mycobacterium tuberculosis growth and enoyl acyl carrier protein reductase (InhA) inhibitors ŞD Doğan, MG Gündüz, H Doğan, VS Krishna, C Lherbet, D Sriram European Journal of Medicinal Chemistry 199, 112402, 2020 | 32 | 2020 |
| Discovery of hydrazone containing thiadiazoles as Mycobacterium tuberculosis growth and enoyl acyl carrier protein reductase (InhA) inhibitors H Doğan, ŞD Doğan, MG Gündüz, VS Krishna, C Lherbet, D Sriram, ... European Journal of Medicinal Chemistry 188, 112035, 2020 | 32 | 2020 |
