Design and synthesis of novel quinoline–aminopiperidine hybrid analogues as Mycobacterium tuberculosis DNA gyraseB inhibitors B Medapi, J Renuka, S Saxena, JP Sridevi, R Medishetti, P Kulkarni, ... Bioorganic & medicinal chemistry 23 (9), 2062-2078, 2015 | 58 | 2015 |
Larval zebrafish model for studying the effects of valproic acid on neurodevelopment: An approach towards modeling autism S Dwivedi, R Medishetti, R Rani, A Sevilimedu, P Kulkarni, P Yogeeswari Journal of pharmacological and toxicological methods 95, 56-65, 2019 | 57 | 2019 |
Novel zebrafish EAE model: A quick in vivo screen for multiple sclerosis P Kulkarni, S Yellanki, R Medishetti, D Sriram, U Saxena, P Yogeeswari Multiple sclerosis and related disorders 11, 32-39, 2017 | 31 | 2017 |
Development of novel N-linked aminopiperidine-based mycobacterial DNA gyrase B inhibitors: scaffold hopping from known antibacterial leads VU Jeankumar, J Renuka, VK Pulla, V Soni, JP Sridevi, P Suryadevara, ... International journal of antimicrobial agents 43 (3), 269-278, 2014 | 31 | 2014 |
Ligand/PTC-free intramolecular Heck reaction: synthesis of pyrroloquinoxalines and their evaluation against PDE4/luciferase/oral cancer cell growth in vitro and zebrafish in vivo PV Babu, S Mukherjee, GS Deora, KS Chennubhotla, R Medisetti, ... Organic & Biomolecular Chemistry 11 (39), 6680-6685, 2013 | 28 | 2013 |
InCl3 mediated heteroarylation of indoles and their derivatization via CH activation strategy: Discovery of 2-(1H-indol-3-yl)-quinoxaline derivatives as a new class of PDE4B … R Sunke, R Bankala, B Thirupataiah, EVVS Ramarao, JS Kumar, ... European Journal of Medicinal Chemistry 174, 198-215, 2019 | 27 | 2019 |
Exploring the gyrase ATPase domain for tailoring newer anti-tubercular drugs: hit to lead optimization of a novel class of thiazole inhibitors VU Jeankumar, S Kotagiri, R Janupally, P Suryadevara, JP Sridevi, ... Bioorganic & Medicinal Chemistry 23 (3), 588-601, 2015 | 26 | 2015 |
Mycobacterium tuberculosis Zinc Metalloprotease-1 Assists Mycobacterial Dissemination in Zebrafish MH Vemula, R Medisetti, R Ganji, K Jakkala, S Sankati, K Chatti, ... Frontiers in Microbiology 7, 1347, 2016 | 21 | 2016 |
NaSH in the construction of thiophene ring fused with N-heterocycles: A rapid and inexpensive synthesis of novel small molecules as potential inducers of apoptosis SK Kolli, A Nakhi, R Medishetti, S Yellanki, P Kulkarni, RR Raju, M Pal Bioorganic & Medicinal Chemistry Letters 24 (18), 4460-4465, 2014 | 21 | 2014 |
Ligand-free MCR for linking quinoxaline framework with a benzimidazole nucleus: a new strategy for the identification of novel hybrid molecules as potential inducers of apoptosis R Sunke, PV Babu, S Yellanki, R Medishetti, P Kulkarni, M Pal Organic & Biomolecular Chemistry 12 (35), 6800-6805, 2014 | 21 | 2014 |
Ruthenium-catalyzed synthesis of pyrrolo [1, 2-a] quinoxaline derivatives from 1-(2-aminophenyl) pyrroles and sulfoxonium ylides XF Cui, FP Hu, XQ Zhou, ZZ Zhan, GS Huang Synlett 31 (12), 1205-1210, 2020 | 19 | 2020 |
Design, Synthesis and Evaluation of 5-pyridin-4-yl-2-thioxo-[1, 3, 4] oxadiazol-3-yl Derivatives as Anti-angiogenic Agents Targeting VEGFR-2 U Bhanushali, S Kalekar-Joshi, R Kulkarni-Munshi, S Yellanki, ... Anti-Cancer Agents in Medicinal Chemistry (Formerly Current Medicinal …, 2017 | 18 | 2017 |
Zebrafish based strategy for the identification of a potential pharmacophore for apoptosis: a greener CuAAC approach for novel 1, 2, 3-triazoles derived from mefenamic acid PV Babu, S Mukherjee, DR Gorja, S Yellanki, R Medisetti, P Kulkarni, ... RSC Advances 4 (10), 4878-4882, 2014 | 18 | 2014 |
PdCl2-catalyzed synthesis of a new class of isocoumarin derivatives containing aminosulfonyl/aminocarboxamide moiety: First identification of a isocoumarin based PDE4 inhibitor B Thirupataiah, G Mounika, GS Reddy, JS Kumar, KA Hossain, ... European Journal of Medicinal Chemistry 221, 113514, 2021 | 16 | 2021 |
Dual drug conjugate loaded nanoparticles for the treatment of cancer M Shyam Matlapudi, A Moin, R Medishetti, K Rajendra, A M Raichur, ... Current drug delivery 12 (6), 782-794, 2015 | 15 | 2015 |
Isovanillin derived N-(un) substituted hydroxylamines possessing an ortho-allylic group: valuable precursors to bioactive N-heterocycles B Dulla, ND Tangellamudi, S Balasubramanian, S Yellanki, R Medishetti, ... Organic & Biomolecular Chemistry 12 (16), 2552-2558, 2014 | 15 | 2014 |
A Pd-based regioselective strategy to indole-1, 2-fused 8-and 9-membered rings: their evaluation as potential scaffolds for apoptosis in zebrafish B Prasad, BY Sreenivas, A Sushma, S Yellanki, R Medisetti, P Kulkarni, ... Organic & Biomolecular Chemistry 12 (18), 2864-2868, 2014 | 14 | 2014 |
PHLPP1 promotes neutral lipid accumulation through AMPK/ChREBP-dependent lipid uptake and fatty acid synthesis pathways K Balamurugan, R Medishetti, J Kotha, P Behera, K Chandra, ... Iscience 25 (2), 2022 | 13 | 2022 |
Rosuvastatin based novel 3-substituted isocoumarins/3-alkylidenephthalides: Ultrasound assisted synthesis and identification of new anticancer agents JS Kumar, B Thirupataiah, R Medishetti, A Ray, SD Bele, KA Hossain, ... European Journal of Medicinal Chemistry 201, 112335, 2020 | 11 | 2020 |
A DNAzyme based knockdown model for Fragile-X syndrome in zebrafish reveals a critical window for therapeutic intervention R Medishetti, R Rani, S Kavati, A Mahilkar, V Akella, U Saxena, P Kulkarni, ... Journal of Pharmacological and Toxicological Methods 101, 106656, 2020 | 11 | 2020 |