Straightforward strategies for the preparation of NH-sulfoximines: a serendipitous story JA Bull, L Degennaro, R Luisi Synlett 28 (19), 2525-2538, 2017 | 129 | 2017 |
Palladium-catalyzed hydroacyloxylation of ynamides DL Smith, WRF Goundry, HW Lam Chemical Communications 48 (10), 1505-1507, 2012 | 103 | 2012 |
Total synthesis of cytotoxic sponge alkaloids hachijodines F and G WRF Goundry, JE Baldwin, V Lee Tetrahedron 59 (10), 1719-1729, 2003 | 67 | 2003 |
Total synthesis of (+)-apiosporamide: assignment of relative and absolute configuration DR Williams, DC Kammler, AF Donnell, WRF Goundry ANGEWANDTE CHEMIE-INTERNATIONAL EDITION IN ENGLISH- 44 (41), 6715, 2005 | 66 | 2005 |
Development of a continuous flow sulfoxide imidation protocol using azide sources under superacidic conditions B Gutmann, P Elsner, A O’Kearney-McMullan, W Goundry, DM Roberge, ... Organic Process Research & Development 19 (8), 1062-1067, 2015 | 60 | 2015 |
Development and scale-up of a biocatalytic process to form a chiral sulfoxide WRF Goundry, B Adams, H Benson, J Demeritt, S McKown, K Mulholland, ... Organic Process Research & Development 21 (1), 107-113, 2017 | 58 | 2017 |
Rhodium-catalyzed [2+ 2] cycloaddition of ynamides with nitroalkenes DL Smith, SR Chidipudi, WR Goundry, HW Lam Organic letters 14 (18), 4934-4937, 2012 | 42 | 2012 |
Development and Scale-up of a Route to ATR Inhibitor AZD6738 WRF Goundry, K Dai, M Gonzalez, D Legg, A O’Kearney-McMullan, ... Organic Process Research & Development 23 (7), 1333-1342, 2019 | 40 | 2019 |
Electrophilic Activation of [1.1. 1] Propellane for the Synthesis of Nitrogen‐Substituted Bicyclo [1.1. 1] pentanes S Livesley, AJ Sterling, CM Robertson, WRF Goundry, JA Morris, F Duarte, ... Angewandte Chemie International Edition 61 (2), e202111291, 2022 | 34 | 2022 |
Late-stage sulfoximidation of electron-rich arenes by photoredox catalysis H Lämmermann, A Sudau, D Rackl, H Weinmann, K Collins, L Wortmann, ... Synlett 29 (20), 2679-2684, 2018 | 26 | 2018 |
Hydrogen‐borrowing Alkylation of 1, 2‐amino Alcohols in the Synthesis of Enantioenriched Γ‐aminobutyric Acids CJJ Hall, WRF Goundry, TJ Donohoe Angewandte Chemie 133 (13), 7057-7061, 2021 | 21 | 2021 |
Synthesis of Sulfur-Substituted Bicyclo [1.1. 1] pentanes by Iodo-Sulfenylation of [1.1. 1] Propellane S Livesley, B Trueman, CM Robertson, WRF Goundry, JA Morris, C Aïssa Organic Letters 24 (38), 7015-7020, 2022 | 16 | 2022 |
C [double bond, length as m-dash] C/B–N substitution in five membered heterocycles. A computational analysis VA Dixit, WRF Goundry, S Tomasi New Journal of Chemistry 41 (9), 3619-3633, 2017 | 15 | 2017 |
An alternative focus for route design for the synthesis of antibody–drug conjugate payloads AC Tiberghien, PW Howard, WRF Goundry, M McCormick, JS Parker The Journal of Organic Chemistry 84 (8), 4830-4836, 2019 | 13 | 2019 |
Total synthesis of cytotoxic sponge alkaloids hachijodines F and G WRF Goundry, V Lee, JE Baldwin Tetrahedron letters 43 (15), 2745-2747, 2002 | 13 | 2002 |
Payloads for antibody–drug conjugates WRF Goundry, JS Parker Organic Process Research & Development 26 (8), 2121-2123, 2022 | 12 | 2022 |
Considerations in the developability of peptides for oral administration when formulated together with transient permeation enhancers S Berg, H Edlund, WRF Goundry, CAS Bergström, NM Davies International journal of pharmaceutics 628, 122238, 2022 | 11 | 2022 |
Extension of hydrogen borrowing alkylation reactions for the total synthesis of (−)-γ-lycorane JJ Christopher, RF William Chemical Communications 58 (32), 4966-4968, 2022 | 11 | 2022 |
Synthesis of excitatory amino acid analogues WRF Goundry, V Lee, JE Baldwin Synlett 2006 (15), 2407-2410, 2006 | 9 | 2006 |
The development of a Dimroth rearrangement route to AZD8931 WRF Goundry, K Boardman, O Cunningham, M Evans, MF Jones, ... Organic Process Research & Development 21 (3), 336-345, 2017 | 7 | 2017 |