Raphael Labruere
Raphael Labruere
Associate professor of Bioorganic Chemistry, Univ. P-Sud
Verified email at u-psud.fr
TitleCited byYear
Self‐Immolative Spacers: Kinetic Aspects, Structure–Property Relationships, and Applications
A Alouane, R Labručre, T Le Saux, F Schmidt, L Jullien
Angewandte Chemie International Edition 54 (26), 7492-7509, 2015
1262015
“Self‐Immolative” Spacer for Uncaging with Fluorescence Reporting
R Labručre, A Alouane, T Le Saux, I Aujard, P Pelupessy, A Gautier, ...
Angewandte Chemie International Edition 51 (37), 9344-9347, 2012
342012
Design, Synthesis, and Biological Evaluation of the First Podophyllotoxin Analogues as Potential Vascular‐Disrupting Agents
R Labručre, B Gautier, M Testud, J Seguin, C Lenoir, S Desbčne‐Finck, ...
ChemMedChem 5 (12), 2016-2025, 2010
262010
Light Activation for the Versatile and Accurate Kinetic Analysis of Disassembly of Self‐Immolative Spacers
A Alouane, R Labručre, T Le Saux, I Aujard, S Dubruille, F Schmidt, ...
Chemistry-A European Journal 19 (35), 11717-11724, 2013
172013
Selbstzerlegende Spacer: kinetische Aspekte, Struktur‐Eigenschafts‐Beziehungen und Anwendungen
A Alouane, R Labručre, T Le Saux, F Schmidt, L Jullien
Angewandte Chemie 127 (26), 7600-7619, 2015
162015
Design and Effective Synthesis of the First 4-Aza-2, 3-didehydropodophyllotoxin Rigid Aminologue: AN-Methyl-4-[(3, 4, 5-trimethoxyphenyl) amino)]-1, 2-dihydroquinoline-lactone
R Labručre, P Helissey, S Desbčne-Finck, S Giorgi-Renault
The Journal of organic chemistry 73 (9), 3642-3645, 2008
162008
Poly (vinyl benzoate) nanoparticles for molecular delivery: Studies on their preparation and in vitro properties
R Labručre, R Sicard, R Cormier, E Turos, L West
Journal of Controlled Release 148 (2), 234-240, 2010
142010
Polyamine-based analogs and conjugates as antikinetoplastid agents
E Jagu, S Pomel, S Pethe, PM Loiseau, R Labručre
European Journal of Medicinal Chemistry 139, 982-1015, 2017
102017
Design, synthesis and in vitro antikinetoplastid evaluation of N-acylated putrescine, spermidine and spermine derivatives
E Jagu, R Djilali, S Pomel, F Ramiandrasoa, S Pethe, R Labručre, ...
Bioorganic & medicinal chemistry letters 25 (2), 207-209, 2015
102015
Synthesis and in vitro antikinetoplastid activity of polyamine–hydroxybenzotriazole conjugates
E Jagu, S Pomel, A Diez-Martinez, F Ramiandrasoa, RL Krauth-Siegel, ...
Bioorganic & medicinal chemistry 25 (1), 84-90, 2017
72017
Disassembly Kinetics of Quinone‐Methide‐Based Self‐Immolative Spacers that Contain Aromatic Nitrogen Heterocycles
A Alouane, R Labručre, KJ Silvestre, T Le Saux, F Schmidt, L Jullien
Chemistry–An Asian Journal 9 (5), 1334-1340, 2014
62014
Efficient syntheses of thiono and dithio analogues of tetronic acid
R Labruere, S Desbčne-Finck, P Helissey, S Giorgi-Renault
Synthesis 2006 (24), 4163-4166, 2006
42006
Attenuating the size and molecular carrier capabilities of polyacrylate nanoparticles by a hydrophobic fluorine effect
R Labručre, E Turos
Bioorganic & medicinal chemistry 20 (16), 5042-5045, 2012
32012
Synthesis and antikinetoplastid evaluation of bis (benzyl) spermidine derivatives
E Jagu, S Pomel, A Diez-Martinez, E Rascol, S Pethe, PM Loiseau, ...
European journal of medicinal chemistry 150, 655-666, 2018
22018
A chemically encoded timer for dual molecular delivery at tailored ranges and concentrations
S Serra, A Alouane, T Le Saux, S Huvelle, R Plasson, F Schmidt, L Jullien, ...
Chemical Communications 54 (49), 6396-6399, 2018
12018
Thienopyrimidinedione Formation Versus Ester Hydrolysis from Ureido Carboxylic Acid Methyl Ester
M Reille-Seroussi, R Labručre, N Inguimbert, S Broussy, N Gagey-Eilstein, ...
Synthesis 45 (04), 479-490, 2013
12013
Synthesis of the 3, 4, 5-Trimethoxy-2-(3, 4-methylenedioxy-6-nitrophenyl) benzaldehyde for Divergent Preparation of Cytotoxic Biaryls
R Labruere, P Helissey, S Desbene-Finck, S Giorgi-Renault
Letters in Organic Chemistry 9 (8), 568, 2012
12012
Arylboronate prodrugs of doxorubicin as promising chemotherapy for pancreatic cancer
C Skarbek, S Serra, H Maslah, E Rascol, R Labručre
Bioorganic chemistry 91, 103158, 2019
2019
Spermine-NBD as fluorescent probe for studies of the polyamine transport system in Leishmania donovani
E Jagu, S Pomel, S Pethe, JC Cintrat, PM Loiseau, R Labručre
Bioorganic & medicinal chemistry letters 29 (14), 1710-1713, 2019
2019
Anti–Methicillin-Resistant Staphylococcus aureus Nanoantibiotics
R Labručre, AJ Sona, E Turos
Frontiers in Pharmacology 10, 2019
2019
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