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Adel Ghiaty
Adel Ghiaty
Professor of organic chemistry
Verified email at azhar.edu.eg
Title
Cited by
Cited by
Year
From triazolophthalazines to triazoloquinazolines: A bioisosterism-guided approach toward the identification of novel PCAF inhibitors with potential anticancer activity
MH El-Shershaby, A Ghiaty, AH Bayoumi, AA Al-Karmalawy, ...
Bioorganic & Medicinal Chemistry 42, 116266, 2021
552021
Investigating the Antibacterial Activity of Biphenylthiazoles against Methicillin- and Vancomycin-Resistant Staphylococcus aureus (MRSA and VRSA)
M Hagras, H Mohammad, MS Mandour, YA Hegazy, A Ghiaty, ...
Journal of Medicinal Chemistry 60 (9), 4074-4085, 2017
462017
Phenylthiazoles with tert-Butyl side chain: Metabolically stable with anti-biofilm activity
A Kotb, NS Abutaleb, MA Seleem, M Hagras, H Mohammad, A Bayoumi, ...
European journal of medicinal chemistry 151, 110-120, 2018
432018
Alkynyl-containing phenylthiazoles: Systemically active antibacterial agents effective against methicillin-resistant Staphylococcus aureus (MRSA)
MM Elsebaei, H Mohammad, M Abouf, NS Abutaleb, YA Hegazy, A Ghiaty, ...
European journal of medicinal chemistry 148, 195-209, 2018
412018
Synthesis and biological evaluation of some [1, 2, 4] triazolo [4, 3-a] quinoxaline derivatives as novel anticonvulsant agents
M Alswah, A Ghiaty, A El-Morsy, K El-Gamal
International Scholarly Research Notices 2013, 2013
412013
1, 2, 4-Triazolo [4, 3-c] quinazolines: a bioisosterism-guided approach towards the development of novel PCAF inhibitors with potential anticancer activity
MH El-Shershaby, A Ghiaty, AH Bayoumi, HEA Ahmed, MS El-Zoghbi, ...
New Journal of Chemistry 45 (25), 11136-11152, 2021
402021
Novel triazolophthalazine-hydrazone hybrids as potential PCAF inhibitors: Design, synthesis, in vitro anticancer evaluation, apoptosis, and molecular docking studies
HS Abulkhair, A Turky, A Ghiaty, HEA Ahmed, AH Bayoumi
Bioorganic Chemistry 100, 103899, 2020
392020
Design, synthesis, and antitumor activity of novel compounds based on 1, 2, 4-triazolophthalazine scaffold: apoptosis-inductive and PCAF-inhibitory effects
A Turky, AH Bayoumi, A Ghiaty, AS El-Azab, AM Alaa, HS Abulkhair
Bioorganic Chemistry 101, 104019, 2020
372020
Synthesis and Evaluation of Some New (1, 2, 4) Triazolo (4, 3‐a) Quinoxalin‐4 (5H)‐one Derivatives as AMPA Receptor Antagonists
H Abul‐Khair, S Elmeligie, A Bayoumi, A Ghiaty, A El‐Morsy, MH Hassan
Journal of Heterocyclic Chemistry 50 (5), 1202-1208, 2013
372013
Design, synthesis, and molecular modelling of pyridazinone and phthalazinone derivatives as protein kinases inhibitors
M Elagawany, MA Ibrahim, HEA Ahmed, AS El-Etrawy, A Ghiaty, ...
Bioorganic & medicinal chemistry letters 23 (7), 2007-2013, 2013
362013
Design, synthesis, and molecular docking studies of new [1,2,4]triazolo[4,3-a]quinoxaline derivatives as potential A2B receptor antagonists
HG Ezzat, AH Bayoumi, FF Sherbiny, AM El-Morsy, A Ghiaty, M Alswah, ...
Molecular Diversity 25, 291-306, 2021
332021
In vivo‐and in silico‐driven identification of novel synthetic quinoxalines as anticonvulsants and AMPA inhibitors
HS Abulkhair, S Elmeligie, A Ghiaty, A El‐Morsy, AH Bayoumi, ...
Archiv der Pharmazie 354 (5), 2000449, 2021
312021
Antimicrobial screening and pharmacokinetic profiling of novel phenyl-[1, 2, 4] triazolo [4, 3-a] quinoxaline analogues targeting DHFR and E. coli DNA gyrase B
AM Omar, M Alswah, HEA Ahmed, AH Bayoumi, KM El-Gamal, A El-Morsy, ...
Bioorganic Chemistry 96, 103656, 2020
282020
Biphenylthiazole antibiotics with an oxadiazole linker: An approach to improve physicochemical properties and oral bioavailability
M Hagras, YA Hegazy, AH Elkabbany, H Mohammad, A Ghiaty, ...
European journal of medicinal chemistry 143, 1448-1456, 2018
282018
4-Substituted benzenesulfonamides featuring cyclic imides moieties exhibit potent and isoform-selective carbonic anhydrase II/IX inhibition
AM Alaa, AS El-Azab, AH Ghiaty, P Gratteri, CT Supuran, A Nocentini
Bioorganic Chemistry 83, 198-204, 2019
252019
Synthesis and evaluation of some new 1, 2, 4-triazolo (4, 3-a) quinoxalin-4-5H-one derivatives as AMPA receptor antagonists
A Bayoumi, A Ghiaty, A El-Morsy, H Abul-Khair, MH Hassan, S Elmeligie
Bulletin of Faculty of Pharmacy, Cairo University 50 (2), 141-146, 2012
222012
tert-Butylphenylthiazoles with an oxadiazole linker: a novel orally bioavailable class of antibiotics exhibiting antibiofilm activity
A Kotb, NS Abutaleb, M Hagras, A Bayoumi, MM Moustafa, A Ghiaty, ...
RSC advances 9 (12), 6770-6778, 2019
182019
Exploration of quinoxaline derivatives as antimicrobial and anticancer agents
AH Bayoumi, AH Ghiaty, SM Abd El‐Gilil, EM Husseiny, MA Ebrahim
Journal of Heterocyclic Chemistry 56 (12), 3215-3235, 2019
152019
Synthesis and biological evaluation of some quinoxaline-2-one derivatives as novel anticonvulsant agents
E Elkaeed, A Ghiaty, A El-Morsy, K El-Gamal, H Sak
Chem Sci Rev Lett 3 (12), 1375-1387, 2014
142014
Azab, AA‐M. Abdel‐Aziz, HS Abulkhair
A Turky, AH Bayoumi, A Ghiaty, AS El
Bioorg. Chem 101, 104019, 2020
92020
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