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Gyanendra Kumar, Ph.D.
Gyanendra Kumar, Ph.D.
Director, Neuron23, Inc
Verified email at neuron23.com - Homepage
Title
Cited by
Cited by
Year
Identification, characterization, and inhibition of Plasmodium falciparum β-hydroxyacyl-acyl carrier protein dehydratase (FabZ)
SK Sharma, M Kapoor, TNC Ramya, S Kumar, G Kumar, R Modak, ...
Journal of Biological Chemistry 278 (46), 45661, 2003
1322003
Discovery of a rhodanine class of compounds as inhibitors of Plasmodium falciparum enoyl-acyl carrier protein reductase
G Kumar, P Parasuraman, SK Sharma, T Banerjee, K Karmodiya, ...
Journal of medicinal chemistry 50 (11), 2665-2675, 2007
1182007
Heterocyclic-Fused Pyrimidines as Novel Tubulin Polymerization Inhibitors Targeting the Colchicine Binding Site: Structural Basis and Anti-Tumor Efficacy.
S Banerjee, KE Arnst, Y Wang, G Kumar, S Deng, L Yang, GB Li, J Yang, ...
Journal of Medicinal Chemistry 61, 1704-1718, 2018
942018
Novel diphenyl ethers: design, docking studies, synthesis and inhibition of enoyl ACP reductase of Plasmodium falciparum and Escherichia coli
M Chhibber, G Kumar, P Parasuraman, TNC Ramya, N Surolia, A Surolia
Bioorganic & medicinal chemistry 14 (23), 8086-8098, 2006
892006
Stable Analogues of OSB‐AMP: Potent Inhibitors of MenE, the o‐Succinylbenzoate‐CoA Synthetase from Bacterial Menaquinone Biosynthesis
X Lu, R Zhou, I Sharma, X Li, G Kumar, S Swaminathan, PJ Tonge, ...
ChemBioChem 13 (1), 129-136, 2012
712012
Green tea catechins potentiate triclosan binding to enoyl-ACP reductase from Plasmodium falciparum (PfENR)
SK Sharma, P Parasuraman, G Kumar, N Surolia, A Surolia
Journal of medicinal chemistry 50 (4), 765-775, 2007
692007
The Structural and Functional Basis for Recurring Sulfa Drug Resistance Mutations in Staphylococcus aureus Dihydropteroate Synthase
E Griffith, M Wallace, Y Wu, G Kumar, S Gajewski, P Jackson, Z Zheng, ...
Front. Microbiol. - Antimicrobials, Resistance and Chemotherapy 9, 2018
652018
Identification of the I38T PA Substitution as a Resistance Marker for Next-Generation Influenza Virus Endonuclease Inhibitors
J Jones, G Kumar, S Barman, I Najera, S White, R Webby, E Govorkova
MBio 9 (2), doi:10.1128/mBio.00430-18, 2018
652018
NMR and molecular modelling studies on the interaction of fluconazole with β-cyclodextrin
SK Upadhyay, G Kumar
Chemistry Central Journal 3, 1-9, 2009
652009
Structure-Guided Design, Synthesis, and Biological Evaluation of (2-(1H-Indol-3-yl)-1H-imidazol-4-yl)(3,4,5-trimethoxyphenyl) Methanone (ABI-231) Analogues Targeting the …
Q Wang, K Arnst, Y Wang, G Kumar, D Ma, SW White, DD Miller, W Li, ...
Journal of Medicinal Chemistry, 2019
632019
A two-helix motif positions the lysophosphatidic acid acyltransferase active site for catalysis within the membrane bilayer
R Robertson, J Yao, S Gajewski, G Kumar, E Martin, C Rock, S White
Nature Structural & Molecular Biology 24, 666-671, 2017
632017
Unfolding studies on soybean agglutinin and concanavalin a tetramers: a comparative account
S Sinha, N Mitra, G Kumar, K Bajaj, A Surolia
Biophysical journal 88 (2), 1300-1310, 2005
632005
N-acylhydrazone inhibitors of influenza virus PA endonuclease with versatile metal binding modes
M Carcelli, D Rogolino, A Gatti, L De Luca, M Sechi, G Kumar, S White, ...
Scientific Reports 6 (31500), 1-14, 2016
572016
Identification and characterization of influenza variants resistant to a viral endonuclease inhibitor
MS Song, G Kumar, WR Shadrick, W Zhou, T Jeevan, Z Li, PJ Slavish, ...
Proceedings of the National Academy of Sciences 113 (13), 3669-3674, 2016
542016
Functional characterization of β-ketoacyl-ACP reductase (FabG) from Plasmodium falciparum
S Pillai, C Rajagopal, M Kapoor, G Kumar, A Gupta, N Surolia
Biochemical and biophysical research communications 303 (1), 387-392, 2003
482003
Unique determinants of neuraminidase inhibitor resistance among N3, N7, and N9 avian influenza viruses
MS Song, BM Marathe, G Kumar, SS Wong, A Rubrum, M Zanin, YK Choi, ...
Journal of virology 89 (21), 10891-10900, 2015
442015
Recent Advances in Computer-Aided Drug Design as Applied to Anti-Influenza Drug Discovery
PL Mallipeddi, G Kumar, SW White, TR Webb
Current Topics in Medicinal Chemistry 14 (16), 1875-1889, 2014
442014
Structural modification of the 3, 4, 5-trimethoxyphenyl moiety in the tubulin inhibitor VERU-111 leads to improved antiproliferative activities
Q Wang, KE Arnst, Y Wang, G Kumar, D Ma, H Chen, Z Wu, J Yang, ...
Journal of medicinal chemistry 61 (17), 7877-7891, 2018
422018
Structure–Activity Relationship Study of Novel 6-Aryl-2-benzoyl-pyridines as Tubulin Polymerization Inhibitors with Potent Antiproliferative Properties
H Chen, S Deng, Y Wang, N Albadari, G Kumar, D Ma, W Li, SW White, ...
Journal of Medicinal Chemistry 63 (2), 827-846, 2020
392020
Combined effect of epigallocatechin gallate and triclosan on enoyl-ACP reductase of Mycobacterium tuberculosis
SK Sharma, G Kumar, M Kapoor, A Surolia
Biochemical and biophysical research communications 368 (1), 12-17, 2008
362008
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