Jayendra Z. Patel
Jayendra Z. Patel
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Diaryl dihydropyrazole-3-carboxamides with significant in vivo antiobesity activity related to CB1 receptor antagonism: Synthesis, biological evaluation, and molecular modeling …
BK Srivastava, A Joharapurkar, S Raval, JZ Patel, R Soni, P Raval, A Gite, ...
Journal of medicinal chemistry 50 (24), 5951-5966, 2007
Chiral 1, 3, 4-oxadiazol-2-ones as highly selective FAAH inhibitors
JZ Patel, T Parkkari, T Laitinen, AA Kaczor, SM Saario, JR Savinainen, ...
Journal of medicinal chemistry 56 (21), 8484-8496, 2013
Biochemical and pharmacological characterization of the human lymphocyte antigen B-associated transcript 5 (BAT5/ABHD16A)
JR Savinainen, JZ Patel, T Parkkari, D Navia-Paldanius, JJT Marjamaa, ...
PLoS One 9 (10), e109869, 2014
Loratadine analogues as MAGL inhibitors
JZ Patel, S Ahenkorah, M Vaara, M Staszewski, Y Adams, T Laitinen, ...
Bioorganic & medicinal chemistry letters 25 (7), 1436-1442, 2015
New in Vitro Tools to Study Human Constitutive Androstane Receptor (CAR) Biology: Discovery and Comparison of Human CAR Inverse Agonists
J Küblbeck, J Jyrkkärinne, F Molnár, T Kuningas, J Patel, ...
Molecular pharmaceutics 8 (6), 2424-2433, 2011
Hair growth stimulator property of thienyl substituted pyrazole carboxamide derivatives as a CB1 receptor antagonist with in vivo antiobesity effect
BK Srivastava, R Soni, JZ Patel, A Joharapurkar, N Sadhwani, ...
Bioorganic & medicinal chemistry letters 19 (9), 2546-2550, 2009
Optimization of 1, 2, 5‐thiadiazole carbamates as potent and selective ABHD6 inhibitors
JZ Patel, TJ Nevalainen, JR Savinainen, Y Adams, T Laitinen, RS Runyon, ...
ChemMedChem 10 (2), 253-265, 2015
Comparative molecular field analysis and molecular dynamics studies of α/β hydrolase domain containing 6 (ABHD6) inhibitors
AA Kaczor, KM Targowska-Duda, JZ Patel, T Laitinen, T Parkkari, ...
Journal of molecular modeling 21, 1-16, 2015
Piperazine and piperidine carboxamides and carbamates as inhibitors of fatty acid amide hydrolase (FAAH) and monoacylglycerol lipase (MAGL)
J Korhonen, A Kuusisto, J van Bruchem, JZ Patel, T Laitinen, ...
Bioorganic & Medicinal Chemistry 22 (23), 6694-6705, 2014
Oxazolidinone antibacterials and our experience
BK Srivastava, R Soni, JZ Patel, MR Jain, PR Patel
Anti-Infective Agents in Medicinal Chemistry (Formerly Current Medicinal …, 2008
Synthesis and in vitro antibacterial activities of novel oxazolidinones
BK Srivastava, MR Jain, M Solanki, R Soni, D Valani, S Gupta, B Mishra, ...
European journal of medicinal chemistry 43 (4), 683-693, 2008
Bioisosteric replacement of dihydropyrazole of 4S-(−)-3-(4-chlorophenyl)-N-methyl-N′-[(4-chlorophenyl)-sulfonyl]-4-phenyl-4, 5-dihydro-1H-pyrazole-1-caboxamidine (SLV-319) a …
BK Srivastava, R Soni, A Joharapurkar, KVVM Sairam, JZ Patel, ...
Bioorganic & medicinal chemistry letters 18 (3), 963-968, 2008
Chemoproteomic, biochemical and pharmacological approaches in the discovery of inhibitors targeting human α/β-hydrolase domain containing 11 (ABHD11)
D Navia-Paldanius, JZ Patel, ML Navarro, H Jakupović, S Goffart, ...
European Journal of Pharmaceutical Sciences 93, 253-263, 2016
1, 3, 4-Oxadiazol-2-ones as fatty-acid amide hydrolase and monoacylglycerol lipase inhibitors: Synthesis, in vitro evaluation and insight into potency and selectivity …
H Käsnänen, A Minkkilä, S Taupila, JZ Patel, T Parkkari, ...
European Journal of Pharmaceutical Sciences 49 (3), 423-433, 2013
Facile synthesis, ex-vivo and in vitro screening of 3-sulfonamide derivative of 5-(4-chlorophenyl)-1-(2, 4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxy lic acid piperidin-1 …
B Kumar Srivastava, R Soni, JZ Patel, S Jha, S Shedage, N Gandhi, ...
Chloroquine fumardiamides as novel quorum sensing inhibitors
M Beus, K Savijoki, JZ Patel, J Yli-Kauhaluoma, A Fallarero, B Zorc
Bioorganic & medicinal chemistry letters 30 (16), 127336, 2020
Strategies to prevent biofilm infections on biomaterials: Effect of novel naturally-derived biofilm inhibitors on a competitive colonization model of titanium by Staphylococcus …
I Reigada, R Pérez-Tanoira, JZ Patel, K Savijoki, J Yli-Kauhaluoma, ...
Microorganisms 8 (3), 345, 2020
Synthesis and in vitro antibacterial activity of novel methylamino piperidinyl oxazolidinones
BK Srivastava, R Soni, JZ Patel, M Solanki, D Valani, S Gupta, B Mishra, ...
Bioorganic & medicinal chemistry letters 17 (18), 5227-5232, 2007
Revisiting 1, 3, 4-oxadiazol-2-ones: utilization in the development of ABHD6 Inhibitors
JZ Patel, J van Bruchem, T Laitinen, AA Kaczor, D Navia-Paldanius, ...
Bioorganic & Medicinal Chemistry 23 (19), 6335-6345, 2015
Docking-based 3D-QSAR studies for 1, 3, 4-oxadiazol-2-one derivatives as FAAH inhibitors
A Zięba, T Laitinen, JZ Patel, A Poso, AA Kaczor
International journal of molecular sciences 22 (11), 6108, 2021
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