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Rodolphe Beaud
Rodolphe Beaud
Senior Scientist, Monte Rosa Therapeutics
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Enantioselective Cu-catalyzed arylation of secondary phosphine oxides with diaryliodonium salts toward the synthesis of P-chiral phosphines
R Beaud, RJ Phipps, MJ Gaunt
Journal of the American Chemical Society 138 (40), 13183-13186, 2016
1622016
FeCl3-mediated Friedel-Crafts hydroarylation with electrophilic N-acetyl indoles for the synthesis of benzofuroindolines.
R Beaud, R Guillot, C Kouklovsky, G Vincent
Angewandte Chemie (International ed. in English) 51 (50), 12546-12550, 2012
1022012
Synthesis of 3-arylated indolines from dearomatization of indoles
N Denizot, T Tomakinian, R Beaud, C Kouklovsky, G Vincent
Tetrahedron letters 56 (30), 4413-4429, 2015
832015
Bioinspired direct access to benzofuroindolines by oxidative [3+ 2] annulation of phenols and indoles
N Denizot, A Pouilhes, M Cucca, R Beaud, R Guillot, C Kouklovsky, ...
Organic letters 16 (21), 5752-5755, 2014
782014
Counteranion-directed catalysis in the Tsuji-Trost reaction: stereocontrolled access to 2, 5-disubstituted 3-hydroxy-tetrahydrofurans.
M Arthuis, R Beaud, V Gandon, E Roulland
Angewandte Chemie (International ed. in English) 51 (42), 10510-10514, 2012
512012
Regioselective Hydroarylation Reactions of C3 Electrophilic N‐Acetylindoles Activated by FeCl3: An Entry to 3‐(Hetero)arylindolines
R Beaud, R Guillot, C Kouklovsky, G Vincent
Chemistry–A European Journal 20 (24), 7492-7500, 2014
472014
Catalyst control over sixfold stereogenicity
X Wu, RM Witzig, R Beaud, C Fischer, D Häussinger, C Sparr
Nature Catalysis 4 (6), 457-462, 2021
382021
Intermolecular dearomative C2-arylation of N-Ac indoles activated by FeCl 3
RK Nandi, F Ratsch, R Beaud, R Guillot, C Kouklovsky, G Vincent
Chemical communications 52 (30), 5328-5331, 2016
372016
Divergent Oxidative Couplings between Indoles and 2, 3-Dihydroxybenzoic Acid Derivatives for the Biomimetic Synthesis of Voacalgine A and Bipleiophylline
N Denizot, D Lachkar, C Kouklovsky, E Poupon, L Evanno, G Vincent
Synthesis 50 (21), 4229-4242, 2018
232018
Triflic Acid as an Efficient Brønsted Acid Promoter for the Umpolung of N‐Ac Indoles in Hydroarylation Reactions
RK Nandi, A Perez‐Luna, D Gori, R Beaud, R Guillot, C Kouklovsky, ...
Advanced Synthesis & Catalysis 360 (1), 161-172, 2018
192018
Revealing the electrophilicity of N-Ac indoles with FeCl 3: a mechanistic study
R Beaud, RK Nandi, A Perez-Luna, R Guillot, D Gori, C Kouklovsky, ...
Chemical Communications 53 (43), 5834-5837, 2017
182017
The quest for an oxidative coupling of phenols and indoles towards benzofuroindolines: a two-stage approach
R Beaud, T Tomakinian, N Denizot, A Pouilhes, C Kouklovsky, G Vincent
Synlett 26 (04), 432-440, 2015
162015
Catalytic carboxylation of heteroaromatic compounds: Double and single carboxylation with CO2
T Mita, H Masutani, S Ishii, Y Sato
Synlett 30 (07), 841-844, 2019
132019
Silver-Mediated Intramolecular Friedel–Crafts-Type Cyclizations of 2-Benzyloxy-3-bromoindolines: Synthesis of Isochromeno [3, 4-b] indolines and 3-Arylindoles
T Yamashiro, K Yamada, H Yoshida, Y Tomisaka, T Nishi, T Abe
Synlett 30 (20), 2247-2252, 2019
92019
Enantioenriched Methylene‐Bridged Benzazocanes Synthesis by Organocatalytic and Superacid Activations
R Beaud, B Michelet, Y Reviriot, A Martin‐Mingot, J Rodriguez, D Bonne, ...
Angewandte Chemie 132 (3), 1295-1301, 2020
82020
N-Iodosuccinimide-Mediated Oxidative Coupling of Indoles and Phenols: A Synthetic Study toward the Benzofuroindoline Moiety of Bipleiophylline
N Denizot, R Guillot, C Kouklovsky, G Vincent
Synthesis 50 (24), 4823-4828, 2018
82018
7-Siloxy-Substituted Hexahydronaphthalene Derivatives: Samarium Diiodide Promoted Synthesis and Typical Reactions
A Niermann, HU Reissig
Synthesis 52 (18), 2721-2730, 2020
52020
Copper-Catalyzed Asymmetric Intermolecular N-Monoarylation of Unprotected Sulfonamides via Desymmetrization of Diaryliodonium Salts at Room Temperature
YL Li, C Zhang, X Jin, XL Yu, Z Wang, HZ Zhang, WQ Yang
Synlett 31 (11), 1077-1081, 2020
32020
Hidden Heptacyclic Chiral N‐Acyl Iminium Ions: A New Entry to Enantioenriched Polycyclic Azepanes and Azocanes by Superacid‐Promoted Intramolecular Pictet …
Y Reviriot, B Michelet, R Beaud, A Martin‐Mingot, F Guégan, ...
Chemistry–A European Journal 28 (25), e202200432, 2022
22022
Publisher Correction: Catalyst control over sixfold stereogenicity
X Wu, RM Witzig, R Beaud, C Fischer, D Häussinger, C Sparr
Nature Catalysis 4 (6), 534-534, 2021
2021
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