Design and synthesis of pyrazole–oxindole conjugates targeting tubulin polymerization as new anticancer agents A Kamal, AB Shaik, N Jain, C Kishor, A Nagabhushana, B Supriya, ... European journal of medicinal chemistry 92, 501-513, 2015 | 113 | 2015 |
Synthesis of β-carboline–benzimidazole conjugates using lanthanum nitrate as a catalyst and their biological evaluation A Kamal, MPN Rao, P Swapna, V Srinivasulu, C Bagul, AB Shaik, ... Organic & Biomolecular Chemistry 12 (15), 2370-2387, 2014 | 69 | 2014 |
The highly selective dopamine D3R antagonist, R-VK4-40 attenuates oxycodone reward and augments analgesia in rodents CJ Jordan, B Humburg, M Rice, GH Bi, ZB You, AB Shaik, J Cao, ... Neuropharmacology 158, 107597, 2019 | 64 | 2019 |
Synthesis, biological evaluation of new oxazolidino-sulfonamides as potential antimicrobial agents A Kamal, P Swapna, RV Shetti, AB Shaik, MPN Rao, S Gupta European Journal of Medicinal Chemistry 62, 661-669, 2013 | 63 | 2013 |
Design and synthesis of imidazo [2, 1-b] thiazole linked triazole conjugates: Microtubule-destabilizing agents SP Shaik, VL Nayak, F Sultana, AVS Rao, AB Shaik, KS Babu, A Kamal European Journal of Medicinal Chemistry 126, 36-51, 2017 | 59 | 2017 |
Synthesis of phenstatin/isocombretastatin–chalcone conjugates as potent tubulin polymerization inhibitors and mitochondrial apoptotic inducers A Kamal, GB Kumar, M Vishnuvardhan, AB Shaik, VS Reddy, R Mahesh, ... Organic & biomolecular chemistry 13 (13), 3963-3981, 2015 | 53 | 2015 |
Design, synthesis and biological evaluation of imidazopyridine/imidazopyrimidine-benzimidazole conjugates as potential anticancer agents A Kamal, GB Kumar, VL Nayak, VS Reddy, AB Shaik, MK Reddy MedChemComm 6 (4), 606-612, 2015 | 53 | 2015 |
Synthesis and biological evaluation of novel pyrano [3, 2-c] carbazole derivatives as anti-tumor agents inducing apoptosis via tubulin polymerization inhibition P Padmaja, GK Rao, A Indrasena, BVS Reddy, N Patel, AB Shaik, ... Organic & biomolecular chemistry 13 (5), 1404-1414, 2015 | 51 | 2015 |
Synthesis of arylpyrazole linked benzimidazole conjugates as potential microtubule disruptors A Kamal, AB Shaik, S Polepalli, GB Kumar, VS Reddy, R Mahesh, ... Bioorganic & medicinal chemistry 23 (5), 1082-1095, 2015 | 50 | 2015 |
Design, synthesis, in silico pharmacokinetics prediction and biological evaluation of 1, 4-dihydroindeno [1, 2-c] pyrazole chalcone as EGFR/Akt pathway inhibitors I Khan, KR Garikapati, A Setti, AB Shaik, VKK Makani, MA Shareef, ... European journal of medicinal chemistry 163, 636-648, 2019 | 45 | 2019 |
Synthesis of (Z)-(arylamino)-pyrazolyl/isoxazolyl-2-propenones as tubulin targeting anticancer agents and apoptotic inducers A Kamal, VS Reddy, AB Shaik, GB Kumar, M Vishnuvardhan, S Polepalli, ... Organic & Biomolecular Chemistry 13 (11), 3416-3431, 2015 | 45 | 2015 |
Synthesis and Biological Evaluation of Imidazopyridine–Oxindole Conjugates as Microtubule‐Targeting Agents A Kamal, VS Reddy, S Karnewar, SS Chourasiya, AB Shaik, GB Kumar, ... ChemMedChem 8 (12), 2015-2025, 2013 | 42 | 2013 |
Pyrazole–oxadiazole conjugates: synthesis, antiproliferative activity and inhibition of tubulin polymerization A Kamal, AB Shaik, S Polepalli, VS Reddy, GB Kumar, S Gupta, ... Organic & Biomolecular Chemistry 12 (40), 7993-8007, 2014 | 41 | 2014 |
Metabolic Profiling and Biological Activities of Bioactive Compounds Produced by Pseudomonas sp. Strain ICTB-745 Isolated from Ladakh,India JJ Ahmed Kamal, Anver Basha Shaik, C. Ganesh Kumar, Poornima Mongolla, P ... J. Microbiol. Biotechnol. (2012), 22 (1), 69–79, 2011 | 41* | 2011 |
Design, synthesis and biological evaluation of 1, 4-dihydro indeno [1, 2-c] pyrazole linked oxindole analogues as potential anticancer agents targeting tubulin and inducing p53 … I Khan, KR Garikapati, AB Shaik, VKK Makani, A Rahim, MA Shareef, ... European Journal of Medicinal Chemistry 144, 104-115, 2018 | 36 | 2018 |
Discovery of pyrrolospirooxindole derivatives as novel cyclin dependent kinase 4 (CDK4) inhibitors by catalyst-free, green approach A Kamal, R Mahesh, VL Nayak, KS Babu, GB Kumar, AB Shaik, ... European Journal of Medicinal Chemistry 108, 476-485, 2016 | 36 | 2016 |
Synthesis of imidazo [2, 1-b][1, 3, 4] thiadiazole–chalcones as apoptosis inducing anticancer agents A Kamal, VS Reddy, K Santosh, GB Kumar, AB Shaik, R Mahesh, ... MedChemComm 5 (11), 1718-1723, 2014 | 33 | 2014 |
Investigation of novel primary and secondary pharmacophores and 3-substitution in the linking chain of a series of highly selective and bitopic dopamine D3 receptor antagonists … AB Shaik, V Kumar, A Bonifazi, AM Guerrero, SL Cemaj, A Gadiano, ... Journal of medicinal chemistry 62 (20), 9061-9077, 2019 | 32 | 2019 |
The Significance of Chirality in Drug Design and Synthesis of Bitopic Ligands as D3 Receptor (D3R) Selective Agonists FO Battiti, SL Cemaj, AM Guerrero, AB Shaik, J Lam, R Rais, BS Slusher, ... Journal of medicinal chemistry 62 (13), 6287-6314, 2019 | 30 | 2019 |
New quinoline linked chalcone and pyrazoline conjugates: Molecular properties prediction, antimicrobial and antitubercular activities NS Rao, AB Shaik, SR Routhu, SMA Hussaini, S Sunkari, AVS Rao, ... ChemistrySelect 2 (10), 2989-2996, 2017 | 30 | 2017 |